ЛАБОРАТОРИЯ
Органического синтеза
НАУЧНО-
ИССЛЕДОВАТЕЛЬСКАЯ
Oxidative Transformation of 2-Furylanilines into Indolin-3-ones
Ekaterina R. Nasibullina, Elena Y. Mendogralo, Anton A. Merkushev, Anton S. Makarov, and Maxim G. Uchuskin. J. Org. Chem. 2024, 89, 9, 6602–6606
Unveiling Orthogonal Reactivity of Substituted 2-(2-Azidostyryl)furans: Thermolysis and Photolysis versus Catalysis
Yury A. Vasev, Ekaterina R. Nasibullina, Anton S. Makarov, and Maxim G. Uchuskin. Org. Lett. 2023, 25, 43, 7780–7785
Mechanistic Insight into Palladium-Catalyzed Asymmetric Alkylation of Indoles with Diazoesters Employing Bipyridine-N,N’-dioxides as Chiral Controllers
Yasuaki Fukazawa, Vladimir Yu. Vaganov, Julia V. Burykina, Artem N. Fakhrutdinov, Ruslan I. Safiullin, Felix Plasser, Aleksandr E. Rubtsov, Valentine P. Ananikov, Andrei V. Malkov. Advanced Synthesis & Catalysis. Volume 366, Issue 1. p. 121-133
Interrupted Furan–Yne Cyclization: Access to Unsaturated Dicarbonyl Compounds and Their Subsequent Transformation into Functionalized Pyridazines
Yury A. Vasev, Ekaterina R. Nasibullina, Anton S. Makarov, and Maxim G. Uchuskin. Org. Lett. 2023, 25, 43, 7780–7785
Synthesis of tetrahydrofuro[3,2-c]pyridines via Pictet–Spengler reaction
Elena Y. Mendogralo and Maxim G. Uchuskin. Beilstein J. Org. Chem. 2023, 19, 991–997
De novo three-component synthesis of meta-substituted anilines
Anton S. Makarov, Arthur N. Bakiev and Diana A. Eshmemeteva. Org. Chem. Front., 2023,10, 2760-2765
Synthetic strategy toward push-pull chromophores on furan-, benzofuran-, pyrrole-, and indole-based matrices
Danil K. Vshivkov, Arthur N. Bakiev, Diana A. Eshmemeteva, Anton S. Makarov
Extended Version of the Corey–Chaykovsky Reaction: Synthesis of 2,4-Substituted Furans by the Treatment of β-Dialkylamino Chalcones with Dimethylsulfonium Methylide
Roman O. Shcherbakov, Danil A. Myasnikov, Igor V. Trushkov, and Maxim G. Uchuskin. Cite this: J. Org. Chem. 2023, 88, 13, 8227–8235
Yi Du, Adelaide Lunga, Aleksandr E. Rubtsov and Andrei V. Malkov.
Green Chemistry. 01 Sep 2022.
Green Chemistry. 01 Sep 2022.
Short Electrochemical Asymmetric Synthesis of (+)-N-Acetylcolchinol
Petrakis N. Chalikidi, Taimuraz T. Magkoev, Andrey V. Gutnov, Oleg P. Demidov, Maxim G. Uchuskin, Igor V. Trushkov, Vladimir T. Abaev. Cite this: J. Org. Chem. 2021, 86, 14, 9838–9846
One-Step Synthesis of Triphenylphosphonium Salts from (Het)arylmethyl Alcohols
Roman O. Shcherbakov, Diana A. Eshmemet’eva, Anton A. Merkushev, Igor V. Trushkov, Maxim G. Uchuskin. Molecules. 2021 May; 26(9): 2637.
Transformation of 3-(Furan-2-yl)-1,3-di(het)arylpropan-1-ones to Prop-2-en-1-ones via Oxidative Furan Dearomatization/2-Ene-1,4,7-triones Cyclization
Anton A. Merkushev, Anton S. Makarov, Pavel M. Shpuntov, Vladimir T. Abaev, Igor V. Trushkov, Maxim G. Uchuskin. European Journal of Organic Chemistry 2021(8)
Oxidative Rearrangement of 2-(2-Aminobenzyl)furans: Synthesis of Functionalized Indoles and Carbazoles
Alexander G Tkachenko, Natalya M Kashevarova, Roman Yu Sidorov, Larisa Yu Nesterova, Anna V Akhova, Ivan V Tsyganov, Vladimir Yu Vaganov, Sergei A Shipilovskikh, Aleksandr E Rubtsov, Andrei V Malkov. Cell Chem Biol. 2021 Feb 9
A synthetic diterpene analogue inhibits mycobacterial persistence and biofilm formation by targeting (p)ppGpp synthetases
Aleksandr E. Rubtsov, Andrei V. Malkov. 2021. Synlett
Developing a Methodology for Catalytic Asymmetric Crotylation of Aldehydes
Aleksandr E. Rubtsov, Andrei V. Malkov. 2021. Synthesis (Germany)
Recent Advances in the Synthesis of 2,2′-Bipyridines and Their Derivatives
Dr. Anton A. Merkushev Dr. Anton S. Makarov Pavel M. Shpuntov Prof. Dr. Vladimir T. Abaev Prof. Dr. Igor V. Trushkov Dr. Maxim G. Uchuskin. European Journal of Organic Chemistry. Volume 2021, Issue 8, 25 February 2021, Pages 1274-1285
Oxidative Rearrangement of 2‐(2‐Aminobenzyl)furans: Synthesis of Functionalized Indoles and Carbazoles
Fukazawa, Y., Rubtsov, A.E., Malkov, A.V. (2020) European Journal of Organic Chemistry, 2020 (22), pp. 3317-3319.
A Mild Method for Electrochemical Reduction of Heterocyclic N‐Oxides
Vaganov, V.Y., Fukazawa, Y., Kondratyev, N.S., Rubtsov, A.E., Malkov, A.V. Advanced Synthesis and Catalysis, 2020, 362(23), стр. 5467–5474
Optimization of Catalyst Structure for Asymmetric Propargylation of Aldehydes with Allenyltrichlorosilane
Shipilovskikh, S.A., Rubtsov, A.E. Russian Journal of General Chemistry, 2020, 90(5), стр. 809–814
Recyclization of 3-(Thiophen-2-yl)imino-3H-furan-2-ones under the Action of Cyanoacetic Acid Derivatives
Zelina, E.Y., Nevolina, T.A., Sorotskaja, L.N., ...Trushkov, I.V., Uchuskin, M.G. Tetrahedron Letters, 2020, 61(9), 151532
Route to pyrrolo[1,2-a]quinoxalines via a furan ring opening-pyrrole ring closure sequence
Shipilovskikh, S.A., Vaganov, V.Y., Makhmudov, R.R., Rubtsov, A.E. Russian Journal of General Chemistry, 2020, 90(4), стр. 583–589
Synthesis and Antinociceptive Activity of N-Substituted 4-Aryl-4-oxo-2-[(3-thiophen-2-yl)amino]but-2-enamides
Fadeev, A.A., Chagarovskiy, A.O., Makarov, A.S., Uchuskin, M.G., Trushkov, I.V. Molecules (Basel, Switzerland), 2020, 25(23)
Synthesis of (Het)aryl 2-(2-hydroxyaryl)cyclopropyl Ketones
Shipilovskikh, S.A., Rubtsov, A.E. Russian Journal of General Chemistry, 2020, 90(6), стр. 943–947
Synthesis of New Substituted 3-(Thien-2-yl)imino-3H-furan-2-ones
